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CYP3A4 activity data at different pre-incubation timees and different concentrations of a time-dependent inhibitor.

Usage

examplinib_in_vitro_tdi

Format

A data frame with 4 columns

  • TIME Pre-incubation time in minutes.

  • CONC Precipitant concentration in uM.

  • ACT Enzyme activity in percent of initial.

  • SOURCE Source study report

Source

Fully synthetic data set to demonstrate TDI-related calculations